Peptide Dermorphin 10mg Vial

Pharmaceutical Strong Effect Peptide Hormone Dermorphin 10mg for Horse

Dermorphin Details:

Product Name: Dermorphin
Alias: Hyp-6
Grade: Pharmaceutical Grade
CAS No: 77614-16-5
Molecular Formula: C40H50N8O10
Molecular Weight: 802.89
Form: Dermorphin ready in 10mg/vial.
Appearance: White powder
Grade: Pharmaceutical Grade
Usage: A strong analgesic
Purity: 99% min
Specification: 5mg/vial; 10mg/vial
Solubility :Distilled water for a solution up to 2 mg/ml

Dermorphin Profile:

Dermorphin Introduction:

1. Dermorphin is a peptide expressed by the frog venom skin glands with a potent opiate-like activity on mu-type opioid receptors, which have potent depressive and analgesic effects. Dermorphin may also have effects on pulmonary ventilation and pituitary hormone release. Dermorphin has been illegally used in horse racing as a performance-enhancing drug. Due to dermorphin’s painkilling activity, horses treated with dermorphin may run harder than they would otherwise.

2. Dermorphin is not found in humans or other mammals and similar D-amino acid peptides have only been found in bacteria, amphibians and molluscs.

3. Dermorphin appears to be made in these through an unusual posttranslational modification carried out by an amino acid isomerase. This unusual process is needed because the D-alanine in this peptide is not among the 20 amino acids coded for in the genetic code and thus the peptide cannot be synthesized in the usual way from the encodings in the genome of an organism.

Dermorphin Usage:

Dermorphin is a hepta-peptide first isolated from the skin of South American frogs belonging to the genus Phyllomedusa. The peptide is a natural opioid that binds as an agonist with high potency and selectivity to mu Opioid receptors.

Dermorphin is about 30-40 times more potent than mor-phine but theoretically may be less likely to produce drug tolerance and addiction (due to its high potency). The amino acid sequence of dermorphin is H-Tyr-D-Ala-Phe-Gly-Tyr-Pro-Ser-NH2.

Dermorphin is a substance that has been demonstrated to act as an agonist at the mu-opiate receptor,” Sams says. “Other mu-opiate agonists are morphinee, fentany, and etorphinee.

We typically associate these substances with analgesic effects in people and dogs, but they produce a paradoxical effect in horses that results in increased locomotor activity at low doses and low blood concentrations.

Peptides and Specification:

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