Procaína Hydrochloride Local Anesthetic Procaine HCl Pó branco 51-05-8
Procaine Hydrochloride Details
Nome do produto: IC de procaina
Alias: Cloridrato de procaína;Aminocaine;Anadolor;Atoxicocaine
Número de registo CAS: 51-05-8
Fórmula molecular: C13H21ClN2O2
Peso molecular: 272.77
Ponto de fusão: 155-156 ° C
Ensaio: 99%
NÚMERO EINECS: 200-077-2
Grau: Qualidade farmacêutica
Armazenamento: Sombreamento, preservação confinada
Aparência: Pó cristalino branco
Especificação de produto:
Nome do produto | IC de procaina |
Número de registro CAS | 51-05-8 |
Aparência | Pó cristalino branco |
Grau | Qualidade farmacêutica |
Pureza | 99%+ Pureza |
Padrão | Empresa padrão |
Quantidade de ordem mínima | 1KG |
Preço | Negociável |
Tipo de aplicativo | Anestésico local |
Outro produto | Benzocaína, Lidocaína, Procaína, Bupivacaína, Tetracaína base |
Aplicação
Procaine HCl is a local anesthetic drug of the amino ester group. It is used primarily to reduce the pain of intramuscular injection of penicillin, and it is also used in dentistry. Owing to the ubiquity of the trade name Novocain, in some regions procaine is referred to generically as novocaine. It acts mainly by being a sodium channel blocker.Today it is used therapeutically in some countries due to its sympatholytic, anti-inflammatory, perfusion enhancing, and mood enhancing effects.
Procaine HCl is indicated for the production of local or regional analgesia and anesthesia by local infiltration and peripheral nerve block techniques.
Benzocaína Uses
Benzocaine is indicated to treat a variety of pain-related conditions. It may be used for:
Local anesthesia of oral and pharyngeal mucous membranes (sore throat, cold sores, mouth ulcers, toothache, sore gums, denture irritation)
Otic pain (earache)
Surgical or procedural local anesthesia
Formulations
Benzocaine can come in a variety of preparations including:
Oral preparations:
Lozenges (ex. Cepacol, Mycinettes)
Topical preparations:
Aerosol (ex. Topex)
Gel (ex. Orajel)
Paste (ex. Orabase)
Benzocaine as API:
Some glycerol-based ear medications for use in removing excess wax as well as relieving ear conditions
such as otitis media and swimmers ear.
Some previous diet products such as Ayds.
Some condoms designed to prevent premature ejaculation. Benzocaine largely inhibits sensitivity on the
penis, and can allow for an erection to be maintained longer (in a continuous act) by delaying ejaculation.
Por outro lado, an erection will also fade faster if stimulus is interrupted
Benzocaine mucoadhesive patches have been used in reducing orthodontic pain.
In Poland it is included, together with menthol and zinc oxide, in the liquid powder (not to be confused with the liquid face powder) used mainly after mosquito stings. Today’s ready made Pudroderm was once used there as pharmaceutical compound.
Benzocaine is commonly found, particularly in Britain, as an impurity in street cocaine and also as a
bulking agent in “legal highs”. Whilst giving a numbing effect similar to cocaine on users’ gums it does not
actually produce the effects of cocaine. Also benzocaine can and has been mistaken for a false positive
for cocaine.
Benzocaine was used in synthesis of Leteprinim.
Vantagem
We have engaged in this line has many years of experience, our reputation is our guarantee of quality. Alta qualidade, competitive price, fast delivery, safe shipping and considerate after-sale service gain the trust and praise from the customers all over the world.
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Our products and services will focus on the largest customer demand, We hold the greatest enthusiasm and sincere cooperation with each customer.
COA
Itens de teste | Especificação de | Resultados do teste |
Aparência | White crystals or a white crystalline powder | Estar em conformidade |
Identificação | ABE. It appears positive reaction |
Ponto de fusão | 154degree~158degree | 154degree~157degree |
Acidity | PH 5.0~6.5 | PH=5.9 |
Aparência da solução | Claro e incolor | Estar em conformidade |
Perda por secagem | ≤ 0.5% | 0.07% |
Metais pesados | ≤0.0005% | Estar em conformidade |
Substâncias afins | ≤0.05% | Estar em conformidade |
Cinzas sulfatadas | 0.1% | 0.05% |
Ensaio ( na base seca ) | 99.0-101.0% | 99.87% |
Conclusão | Conform to BP2005 |
Pó de anestésico local:
Articaína | Fluoresceína HCL |
Articaína HCl | Novocaína HCL |
Benzocaína | Prilocaína |
Benzocaína HCL | Procaína |
Bupivacaína | Procaína HCL |
Bupivacaína HCL | Cloridrato de procaína |
Cloridrato de Dibucaína | Cloridrato de Proparacaine |
Dimethocaine HCL | Propitocaine |
Cloridrato de Dyclonine | Cloridrato de Propitocaine |
Epinefrina | Mesilato de ropivacaína |
Epinefrina HCL | Tetracaína |
Cloridrato de levobupivacaína | Base de tetracaína |
Lidocaína | Tetracaína HCL |
Lidocaína HCL | Cloridrato de tetracaína |
Cloridrato de lidocaína | |
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